Bremelanotide · Vyleesi · PT141

PT-141 (Bremelanotide): research profile.

Melanocortin receptor agonist studied for sexual function and libido research. FDA-approved as Vyleesi for hypoactive sexual desire disorder in premenopausal women.

peptide
Category
~2.7 hours
Half-life
human_trials
Status
Human TrialsBremelanotide · Vyleesi · PT141

Properties

Category
peptide
Molecular weight
1025.2 g/mol
Half-life
~2.7 hours
Storage
2-8°C reconstituted
CAS number
189691-06-3

Mechanism

Non-selective melanocortin receptor agonist (MC1R-MC5R) with primary activity at MC3R and MC4R. Acts centrally on neural pathways controlling sexual arousal.

Research sourcing

For research purposes only
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Primary research

Read what the peer-reviewed literature actually says about PT-141 (Bremelanotide) directly on PubMed.

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